DiePharmazie 4/2001




Abdel-Rahman, R. M.: Chemistry of uncondensed 1,2,4-triazines, part IV. Synthesis and chemistry of bioactive 3-amino-1,2,4-triazines and related compounds – an overview


Original articles

Laszlovszky, I.; Ács, T.; Kiss, B.; Domány, G.Y.: Substituted phenoxyalkylpiperazines as dopamine D3 receptor ligands

Bielawska, A.; Chrzanowski, K.; Bielawski, K.; Palka, J.: Decreased cytotoxicity and increased antimitotic activity of a proline analogue of chlorambucil as a prodrug susceptible to the action of fibroblast’s prolidase

Gobec, S.; Urleb, U.; Auger, G.; Blanot, D.: Synthesis and biochemical evaluation of some novel N-acyl phosphono- and phosphinoalanine derivatives as potential inhibitors of the d-glutamic acid-adding enzyme

Saraç, S.; Yarim, M.; Ertan, M.; Kiliç, F. S.; Erol, K.: 4-Aryl-6,6-dimethyl-1,2,3,4,5,6,7,8-octahydroquinazoline-2,5-diones: synthesis, chromatographic resolution and pharmacological activity

Görlitzer, K.; Wichers, M.; Jones, P. G.: Unexpected formation of spiro[benzofuran-2,2’-[1,4]benzothiazines] from aurones (in German)

Hess, S.; Dölker, M.; Haferburg, D.; Kertscher, H. P.; Matysik, F.-M.; Ortwein, J.; Teubert, U.; Zimmermann, W.; Eger, K.: Separation, analysis and syntheses of trimethoprim impurities

Binsumait, I. A.; Hadidi, K. A.; Abu-Al Raghib, S.: Stability of fluoxetine in stored plasma, aqueous, and methanolic solutions determined by HPLC with UV detection

Hanna, G. M.: Direct enantiomeric purity determination of the chiral anesthetic drug bupivacaine by 1H NMR spectroscopy

Scalia, S.; Simeoni, S.; Bousquet, E.: Determination of bronopol in cosmetic products by HPLC with electrochemical detection

Zaghloul, A. A.; Faltinek, J.; Vaithiyalingam, S. R.; Reddy, I. K.; Khan, M. A.: Naproxen-Eudragit microspheres: screening of process and formulation variables for the preparation of extended release tablets

Klinger, G.; Piater, T.; Jäger, R.; Küntzel, B.; Schön, R.; Hobe, G.: Non-protein dienogest in serum and salivary dienogest in women taking the oral contraceptives Certostat® and Valette®

Mühlenfeld, K.; Langner, A.: Cytochrome P450 1A1 and 4A activities in isolated rat spleen lymphocytes

Jamie, H.; Dyason, K.; Milne, P. J.; Grant, G.; Graz, C. M. J.: The influence of acetoacetate and butyrate on calcium influx and ATP concentrations in HT-29 cells

Tannergren, C.; Langguth, P.; Hoffmann, K.-J.: Compound mixtures in Caco-2 cell permeability screens as a means to increase screening capacity

Schnitzler, P.; Schön, K.; Reichling, J.: Antiviral activity of Australian tea tree oil and eucalyptus oil against herpes simplex virus in cell culture

Michael, H.N.; Salib, J. Y.; Ishak, M. S.: New methoxyflavone glycosides from Verbena bipinnatifida Nutt.