DiePharmazie 5/2005

Original articles


Kettler K, Sakowski J, Wiesner J, Ortmann R, Jomaa H, Schlitzer M: Novel lead structures for antimalarial farnesyltransferase inhibitors

Elmegeed GA, Wardakhan WW, Baiuomy AR: Synthesis of thiazolyl and thieno cholestane derivatives: a novel class of potent anti-inflammatory steroids

Xiaoyan Chen, Feng Qiu, Dafang Zhong, Xiaotao Duan, Changxiao Liu: Validated liquid chromatography-tandem mass spectrometric method for the quantitative determination of daidzein and its main metabolite daidzein glucuronide in rat plasma

Wagner KG, Dowe U, Zadnik J: Highly loaded interactive mixtures for dry powder inhalers: Prediction of the adhesion capacity using surface energy and solubility parameters

Mbah CJ: Effect of electrolytes on the partition coefficient of irbesartan

Chavanpatil MD, Vavia PR: Nasal drug delivery of sumatriptan succinate

Hoffmann C, Müller-Goymann CC: Use of artificial skin constructs in permeation studies of clindamycin phosphate

Fu XC, Song ZF, Fu CY, Liang WQ: A simple predictive model for blood-brain barrier penetration

Merschman SA, Rose MJ, Pearce GES, Woolf EJ, Schaefer BH, Huber AC, Musson DG, Petty KJ, Rush DJ, Varsolona RJ, Matuszewski BK: Characterization of the solubility of a poorly soluble hydroxylated metabolite in human urine and its implications for potential renal toxicity

Vargas F, Rivas C, Perdomo H, Rivas A, Ojeda LE, Velásquez M, Correia H, Hernández A, Fraile G: Clozapine prevents apoptosis and enhances receptor-dependent respiratory burst in human neutrophils

Goel RK, Thind JS, Bal CS, Mahajan MP, Kulkarni SK: Hypocholesterolemic activity of some novel azetidin-2-ones in diet and diabetes induced hypercholesterolemia in rats

Pei-Han Xu, Qiang Cheng, Hong-Fang Li, Ye Yu, Xiang Yan, Rui Wang: The relaxant effect of dobutamine on porcine coronary arterial ring segments

Qi Zhang, Jing Pan, Rong-Liang Zheng, Qin Wang: Redifferentiation of human hepatoma cell induced by 6-(p-chlorophenyl)-3-[1-(p-chlorophenyl)-5-methyl-1H-1,2,3-triazol-4-yl]-
s-triazolo[3,4-b]-1,3,4-thiadiazole (TDZ)

Sathish Sekar D, Sivagnanam K, Subramanian S: Antidiabetic activity of Momordica charantia seeds on streptozotocin induced diabetic rats

Hinrikus T, Tankler H, Raal A: PhD theses at the university of Tartu/Dorpat supervised by Georg Dragendorff 1864-1894 (in German)


Short communications

De Souza AO, Pedrosa MTC, Alderete JB, Cruz AF, Prado MAF, Alves RB, Silva CL: Cytotoxicity, antitumoral and antimycobacterial activity of tetrazole and oxadiazole derivatives

Umadevi S, Mohanta GP, Manavalan R: Studies on antipyretic and anti-inflammatory activities of Scaevola frutescens