DiePharmazie 6/2006



Sharma S, Kulkarni J, Pawar AP: Permeation enhancers in the transmucosal delivery of macromolecules


Original articles

Rizzetto E, Castellano S, Florio C, Vadori M, Stefancich G: 5-Aryl-imidazo[2,1-c][1,4]benzodiazepine derivatives as tricyclic constrained analogues of diazepam and Ro5-4864. Synthesis and binding properties at peripheral and central benzodiazepine receptors

Manolov I, Machulla HJ, Momekov G: Synthesis, physicochemical characterization and preliminary pharmacological in vitro evaluation of two novel cytotoxic benzophenone-linked 3,3-dimethyltriazenes

Liszkiewicz H, Kowalska MW, Rutkowska M, Gliniak H: Synthesis and anxiolytic activity of 1-phenyl-2-(4-aryl-1,3,4,5- tetrahydropyrido[2,3-b][1,4]diazepin-2-ylidene)-ethanone

Szabó Gy, Fischer J, Kis-Varga Ŕ: Synthesis of the pyrazole isostere of valdecoxib

Chavanpatil MD, Rajeshkumar NV, Gulati A: Determination of endothelin antagonist, BMS182874 in plasma by high-performance liquid chromatography

Netriova J, Blahova E, Johanesova Z, Brandsteterova E, Lehotay J, Serdt K, Mocak J: HPLC determination of morphine, morphine-3-glucuronide and morphine-6-glucuronide in human serum of oncological patients after administration of morphine drugs

Mikiciuk-Olasik E, Bilichowski I, Wojewoda E, Witczak M: HPLC method for determination of the purity of a mebrofenin-ligand for 99mTc-complexes l

Weyhers H, Ehlers S, Hahn H, Souto EB, Müller RH: Solid Lipid Nanoparticles (SLN) - Effects of lipid composition on in vitro degradation and in vivo toxicity

De Spiegeleer B, Wattyn E, Slegers G, Veys P, Derrieu G, Van Vooren L: Characterisation of a preservative system in an oily preparation

Bartošíková L, Necas J, Suchý V, Janoštíková E, Bartošík T, Jurica J, Florian T, Klusáková J, Frydrych M: Protective effects of osajin in ischemia-reperfusion of laboratory rat kidney

Wei-Dong Xie, Xue Gao, Tang Shen, Zhong-Jian Jia: Two new benzofurans and other constituents from Ligularia przewalskii

Wiedenfeld H, Montes C, Tawil B, Contin A, Wynsma R: Pyrrolizidine alkaloid level in Senecio bicolor (Willd.) Tod, ssp. cineraria (DC.) from Middle Europe


Short communications

Jha A, Dimmock JR: 1-N-(Arylmaleamoyl)3,5-bis(phenylmethylene)-4- piperidones: a novel class of antimycobacterial agents

Másson M, Benediktsson T, Thorsteinsson T., Loftsson T: Investigation of soft long chain quaternary ammonium compounds as co-factors to enhance in vitro gene delivery

Tomic MA, Vuckovic SM, Stepanovic-Petrovic RM, Ugrešic N, Prostran MŠ, Boškovic B: Peripheral anti-hyperalgesia by oxcarbazepine: involvement of adenosine A1 receptors

Kuželová M, Mladonická M, Bukovský M, Dubnicková M, Adameová A, Švec P: NO-synthase inhibitors provide influence on protective effect of modified endotoxine diphosphoryl lipid A in a rat heart model of ischemic-reperfusion injury

Thuy TT, Sung TV, Hao NT: An eudesmane glycoside from Fissistigma pallens