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CONTENTS
DiePharmazie 06/1997

Original Articles

Stark, H.; Ligneau, X.; Lipp, R.; Arrang, J.-M.; Schwartz, J.-C.; Schunack, W.: Search for novel leads for histamine H3-receptor antagonists: amine derivatives

Mokrosz, M. J.; Mokrosz, J. L.; Duszynska, B.; Deren-Wesolek, A.; Klodzinska, A.; Kowalski, P.; Charakchieva-Minol, S.; Tatarczynska, E.; Kowalska, T.; Majka, Z.; Chojnacka-Wójcik, E.; Misztal, S.: 5-HT1A and 5-HT2A receptor affinity and functional profile of some N-[3-(4-Aryl-1-piperazinyl)propyl] derivatives of indolin-2(1H)-one, quinolin-2(1H)-one and isoquinolin-1(2H)-one

Dannhardt, G.; Kreher, M.; Nowe, U.; Schmitt, S.: 2-Aryl-pyrrolo[2,1-b]benzothiazoles as selective or dual inhibitors of the cyclooxygenase and the 5-lipoxygenase. Non-steroidal antiinflammatory agents, part 21 (in German)

Geies, A. A.; Kamal El-Dean, A. M.; Moustafa, O. Sh.: Synthesis of new triazoloquinoxalines, pyrroloquinoxalines and pyrimidopyrroloquinoxalines

Stamm, H.; Baumann, T.: Synthesis of the first -ylidene--amidobutyronitriles

Rath, S.; Hoffmann, H.: Mechanism of the polarographic reduction of 5-bromo-5-nitro-1,3-dioxane (Bronidox reg.)

Klimes, J.; Mokry, M.: High performance liquid chromatographic analysis of selected sulfonamides in plasma

Michelitsch, A.; Zellnig, K.; Baumeister, A.; Schubert-Zsilavecz, M.; Likussar, W.: Determination of chimaphilin in Chimaphila imbellata primary tincture by differential pulse polarography (in German)

Pérez-Barrales, M. J.; Caraballo, J.; Rabasco, A. M.: Kinetic study of thiomersal degradation products

Thoma, K.; Kübler, N.; Reimann, E.: Photodegradation of antimycotic drugs 4. Communication: Photodegradation of flucytosine and griseofulvin (in German)

Loftsson, T.; Seir Petersen, D.; Le Goffic, F.; Olafsson, J. H.: Unsaturated glycerol monoethers as novel skin penetration enhancers

Diaz, L. M.; Cal, S.; Souto, S.; Concheiro, A.; Gomez-Amoza, J. L.; Martinez-Pacheco, R.: Eudragit RS as major excipient in controlled release tablets for plant dry extracts

Adel, M. S.; Geneidi, A. S.; Ali Shoukri, R.; Saad, I.: In vitro evaluation of flutamide-carrier systems,part 2: Preparation and evaluation of flutamide systems with -cyclodextrin and ß-cyclodextrin

Ahmed, M.; Sadhu, S. K.; Datta, B. K.; Kundu, J.; Bachar, S. C.: Preliminary studies on the antiinflammatory, analgesic and diuretic activity of stagninol, a sesquiterpene isolated from Persicaria stagnina

Schimmer, O.; Eschelbach, H.: Esculetin in Alchemilla speciosa: identification and antimutagenic properties


Short communications


Leibrock, J.; Prücher, H.; Rautenberg, W.: EMD 95885, a new eliprodil analogue with higher affinity for the N-methyl-D-aspartate (NMDA) receptor

Beyer, U.; Schumacher, P.; Unger, C.; Frahm, A. W., Kratz, F.: Synthesis of maleimide derivatives of the anticancer drugs 5-fluorouracil and 5'-deoxy-5-fluorouridine for the preparation of chemoimmunoconjugates

Merkle, S.; Otto, H.-H.: Properties and reactions of substituted 1,2-thiazetidine 1,1-dioxides: about the reaction of 3-acetoxy 1,2-thiazetidine 1,1-dioxide with N-nucleophiles

Radwan, Sh. M.; Kamal El-Dean, A. M.: Pyridazine derivatives: Synthesis and reactions of some new indenol[1,2-d] pyridazine derivatives

Coskun, N. Y.; Aycan, S.; Sungur, S.: Differential pulse polarographic determination of pravastatin sodium in tablets

Narsai, K.; De Villiers, M. M.; Du Plessis, J. : The effect of a change in ionic character on the rheological properties of stearate type O/W creams containing -hydroxy acids

Celková, H.; Sedlárová, E.; Cizmárik:, J.: Relationship between the structure of some 1,4-piperazine derivatives of aryloxyaminopropanols and their Ca-antagonistic activity

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