DiePharmazie 10/2004


Original articles

Obreza, A. ; Stegnar, M. ; Trampuš-Bakija ; Preželj, A. ; Urleb, U. : Synthesis and in vitro evaluation of new azaphenylalanine derivatives as serine protease inhibitors

Fucik, K.; Kettler, K.; Wiesner, J.; Ortmann, R.; Unterreitmeier, D.; Krauss, J.; Bracher, F.; Jomaa, H.; Schlitzer, M.: 2-(Arylpropionylamino)- and 2(arylacryloylamino)benzophenones: Farnesyltransferase inhibition and antimalarial activity

Alagarsamy, V.: Synthesis and pharmacological investigation of some novel 2-methyl-3-(substituted  methylamino)-(3H)-quinazolin-4-ones as histamine H1-receptor blockers

Pískala, A.; Vachálková, A.; Masojídková, M.; Horváthová, K.; Ovesná, Z.; Paces, V.; Novotný, L.: Improved synthesis, antibacterial activity and potential carcinogenicity of 5-amino-1,2,4-thiadiazol- 3(2H)-one

Görlitzer, K.; Lorenz, A.: Medium sized rings from alprenolol and oxprenolol (in German)  

Demirci, B.; Goppel, M.; Demirci, F.; Franz, G.: HPLC profiling and quantification of active principles in leaves of Hedera helix L.

Agrawal, S.; Panchagnula R.: In vitro analysis of rifampicin and its effect on quality control tests of rifampicin containing dosage forms 

Agrawal, S.; Panchagnula, R.: In vitro evaluation of fixed dose combination tablets of anti-tuberculosis drugs after real time storage at ambient conditions 

Di Mambro, V. M.; Maia Campos, P. M. B. G.; Fonseca, M. J. V.: Physical and chemical stability of different formulations with superoxide dismutase  

Xun Sun; Fang Wu; Wei Lu; Zhi-Rong Zhang: Sustained-release hydroxycamptothecin polybutylcyanoacrylate nanoparticles as a liver targeting drug delivery system

Kuca, K.; Cabal, J.; Kassa, J.: A comparison of the efficacy of a bispyridinium oxime – 1,4-bis-(2-hydroxyiminomethylpyridinium) butane dibromide and currently used oximes to reactivate sarin, tabun of cyclosarin-inhibited acetylcholinesterase by in vitro methods

Hamdan, I. I.; Afifi, F.; Taha, M. O.: In vitro alpha amylase inhibitory effect of some clinically-used drugs 

Chun-Ming Wang; Hua Yang; Ya-Ming Wei; Zhon-Jian Jia; Rong-Liang Zheng: In vitro effects on proliferation, telomerase activity and apoptosis of an eremophilanoid sesquiterpene from Senecio oldhamianus Maxim in cultured human tumor cell lines

Ai-Xia Wang; Qi Zhang; Zhong-Jian Jia: A new furobenzopyranone and other constituents from Anaphalis lactea


Short communications

Shah, S. P.; Misra, A.: Liposomal Amphotericin B dry powder inhaler: Effect of fines on in vitro performance

Sznitowska, M.; Pietkiewicz, J.; Stokrocka, M.; Janicki, S.: Dissolution test for ivermectin in oral veterinary paste

Xiang Mei Wu; Pengfei Tu: Chemical properties of a mannoglucan from Cistanche deserticola